Paper I
2022 February (2019 Scheme) · 100 marks · 180 min

Question

Enumerate Alpha blockers and explain their therapeutic uses. (1+3)

Q104 marksShort Answers

Answer

Alpha blockers: Prazosin, Terazosin, Doxazosin (alpha-1 selective); Phenoxybenzamine (non-selective, irreversible); Tamsulosin (alpha-1A selective, uroselective).

Therapeutic uses:

  • Hypertension — Prazosin/Terazosin/Doxazosin reduce peripheral resistance by blocking vascular alpha-1 receptors.
  • Benign prostatic hyperplasia — Tamsulosin relaxes bladder neck/prostatic smooth muscle (alpha-1A selectivity minimizes vascular/hypotensive effects), relieving obstructive urinary symptoms.
  • Pheochromocytoma — Phenoxybenzamine, given pre-operatively to control catecholamine-driven hypertension before tumour resection.

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